Medicine Overview

Indication

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Adult Dose

Clinical InformationAdministration Information
Indication: Adjuvant treatment of Stage III colon cancer
Age: Adult
Condition: Single agent
Dose: Oral – 1,250 mg/m2
Frequency: twice daily
Duration: first 14 days of each 21-day cycle for a maximum of 8 cycles
Indication: Adjuvant treatment of Stage III colon cancer
Age: Adult
Condition: In combination with oxaliplatin-containing regimens
Dose: Oral – 1,000 mg/m2
Frequency: twice daily
Duration: first 14 days of each 21-day cycle for a maximum of 8 cycles
Note: In combination with oxaliplatin 130 mg/m2 administered intravenously on day 1 of each cycle

Child Dose

Clinical InformationAdministration Information
Age: Child
Dose: No approved pediatric dosage available
Note: No approved pediatric dosage available

Renal Dose

Clinical InformationAdministration Information
Condition: Mild renal impairment (Creatinine Clearance 51-80 mL/minute)
Dose: Not mentioned
Note: No dose reduction necessary
Condition: Moderate renal impairment (Creatinine Clearance 30-50 mL/minute)
Dose: Not mentioned – 950 mg/m2
Frequency: twice daily
Note: Reduce dose to 75% of starting dose (ie, from 1250 mg/m2 to 950 mg/m2 twice daily)
Administration
  • Take with food
  • Take within 30 minutes after meal
Side Effect

Drug Interaction

Drug NameRisk Factors
Antacids containing aluminum and magnesium
Drug interaction reported
Leucovorin, Anticoagulants (Warfarin, Heparin, Dabigatran, Rivaroxaban, Apixaban, Edoxaban), phenytoin, allopurinol
Drug interaction reported

Disease Interaction

Disease NameRisk Factors
Severe Renal Impairment
Can cause severe toxicity in patients with kidney dysfunction

Pregnancy

Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage
Product should be stored at a dry place of controlled room temperature below 30° C and kept out of the reach of children.

Data Sources

Clinical & regulatory information on this page is compiled from the following government sources:

DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.