Medicine Overview

Indication

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Adult Dose

Clinical InformationAdministration Information
Indication: Assisted reproductive technologies
Age: Adult
Dose: Subcutaneous Injection – 0.25 mg
Frequency: once daily
Duration: until ovulation induction
Note: As acetate; administered either in the morning beginning on day 5 or 6 of ovarian stimulation or in the evening beginning on day 5.
Indication: Infertility Treatment
Condition: Inhibition of premature LH surges in women undergoing controlled ovarian stimulation
Dose: Subcutaneous Injection – 0.25 mg
Frequency: once daily
Duration: until day of human chorionic gonadotropin administration
Note: Initiate cetrorelix 0.25 mg subcutaneously once daily during early- to mid-follicular phase. Cetrotide 0.25 mg administered on either stimulation day 5 (morning or evening) or day 6 (morning).

Child Dose

Clinical InformationAdministration Information
Age: Child
Dose: Safety and efficacy not established
Note: Safety and efficacy not established

Renal Dose

Clinical InformationAdministration Information
Condition: Mild-to-moderate renal impairment
Dose: Dosage Form – Not specified
Note: Dose adjustment not described by manufacturer
Condition: Severe renal impairment
Dose: Dosage Form – Not specified
Note: Contraindicated
Administration
  • For subcutaneous injection only
  • Follow exact timing as prescribed
Side Effect

Drug Interaction

Drug NameRisk Factors
No specific interactions listed, but possibility of interactions with commonly used medicinal products cannot be entirely excluded
-

Disease Interaction

Disease NameRisk Factors
Moderate to Severe Renal Impairment
Risk of drug accumulation
Moderate to Severe Hepatic Impairment
Risk of drug toxicity

Pregnancy

Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage
Store cetrorelix acetate at room temperature, between 15 to 30° C

Data Sources

Clinical & regulatory information on this page is compiled from the following government sources:

DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.