Medicine Overview

Indication

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Adult Dose

Clinical InformationAdministration Information
Indication: Mantle Cell Lymphoma
Condition: Previously untreated
Dose: Intravenous Injection – 1.3 mg/m²
Frequency: twice weekly for 2 weeks (days 1, 4, 8, 11) followed by a 10-day rest period (days 12 to 21)
Duration: six 3-week cycles; may continue for 8 cycles if the response is first seen at cycle 6
Note: Give with rituximab 375 mg/m² intravenous, cyclophosphamide 750 mg/m² intravenous, and doxorubicin 50 mg/m² intravenous on day 1, plus prednisone 100 mg/m² intravenous on days 1-5
Indication: Mantle Cell Lymphoma
Condition: Relapsed
Dose: Intravenous or Subcutaneous Injection – 1.3 mg/m²/dose
Frequency: twice weekly for 2 weeks (days 1, 4, 8, 11) followed by a 10-day rest period (days 12 to 21)
Note: Therapy extending beyond 8 cycles: Give standard schedule

Child Dose

Clinical InformationAdministration Information
Age: Pediatric
Dose: Not applicable – No approved pediatric dosage available
Note: No approved pediatric dosage available

Renal Dose

Clinical InformationAdministration Information
Condition: Renal Impairment
Dose: Injection – No starting dosage adjustment recommended
Note: In patients requiring dialysis, Bortezomib Injection should be administered after the dialysis procedure
Administration
  • Given as IV or subcutaneous injection
  • Must be administered by healthcare professionals
Side Effect

Drug Interaction

Drug NameRisk Factors
Amiodarone, Antivirals (Acyclovir, Valacyclovir, Ganciclovir, Ribavirin), isoniazid, nitrofurantoin, Statins (Atorvastatin, Simvastatin, Rosuvastatin, Pravastatin, Lovastatin, Fluvastatin)
Concurrent use may increase the chance of peripheral neuropathy
Antihypertensive (Captopril, Enalapril, Lisinopril, Ramipril, Benazepril, Fosinopril, Quinapril, Perindopril, Losartan, Valsartan, Candesartan, Irbesartan, Telmisartan, Olmesartan, Propranolol, Metoprolol, Atenolol, Carvedilol, Bisoprolol, Nadolol, Amlodipine, Diltiazem, Verapamil, Nifedipine, Nicardipine, Hydrochlorothiazide, Chlorthalidone, Indapamide, Furosemide, Bumetanide, Torsemide, Spironolactone, Amiloride, Triamterene, Prazosin, Doxazosin, Terazosin, Clonidine, Methyldopa, Hydralazine, Minoxidil)
Concurrent use increases the chance of hypotension

Disease Interaction

Disease NameRisk Factors
Hypersensitivity
Can cause severe allergic reactions

Pregnancy

Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage
Unopened vials may be stored at controlled room temperature 25º C

Data Sources

Clinical & regulatory information on this page is compiled from the following government sources:

DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.