Medicine Overview

Indication

Know Medicine, Follow Guideline

Adult Dose

Clinical InformationAdministration Information
Indication: Heart Failure Risk Reduction
Age: Adults
Condition: Symptomatic chronic heart failure and ejection fraction less than 45%, following hospitalization for heart failure or need for outpatient intravenous diuretics
Dose: by mouth – 2.5 mg
Frequency: once daily
Note: Initial dose
Indication: Heart Failure Risk Reduction
Age: Adults
Condition: Symptomatic chronic heart failure and ejection fraction less than 45%, following hospitalization for heart failure or need for outpatient intravenous diuretics
Dose: by mouth – 10 mg
Frequency: once daily
Note: Maintenance dose; double dose every 2 weeks as tolerated to target dose

Child Dose

Clinical InformationAdministration Information
Age: Pediatric
Dose: Form – No approved pediatric dosage available
Note: No approved pediatric dosage available

Renal Dose

Clinical InformationAdministration Information
Age: Adult
Condition: eGFR greater than 15 mL/min/1.73m2 and not on dialysis
Dose: Not specified – Not specified
Note: No dosage adjustment necessary
Age: Adult
Condition: eGFR less than 15 mL/min/1.73m2 or on dialysis
Dose: Not specified – Not specified
Note: Not studied
Administration
  • Should be taken with food
  • Take at same time each day
Side Effect

Drug Interaction

Drug NameRisk Factors
Other sGC Stimulators (Soluble Guanylate Cyclase Stimulators)
Coadministration is contraindicated
PDE-5 inhibitors
Coadministration not recommended due to potential for hypotension

Disease Interaction

Disease NameRisk Factors
No specific contraindications listed
Monitor for general drug reactions

Pregnancy

Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage

Details coming soon

Data Sources

Clinical & regulatory information on this page is compiled from the following government sources:

DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.