Medicine Overview

Indication

Know Medicine, Follow Guideline

Adult Dose

Clinical InformationAdministration Information
Indication: Anxiety
Age: Adult
Dose: Tablet – 2-10 mg
Frequency: by mouth every 6-12 hours
Note: No more than 30 mg per 8 hours
Indication: Anxiety
Age: Adult
Dose: Injection – 2-10 mg
Frequency: intravenous or intramuscular every 6-12 hours
Note: No more than 30 mg per 8 hours

Child Dose

Clinical InformationAdministration Information
Indication: Sedative/Muscle Relaxant
Age: less than 6 months
Dose: Not recommended
Note: Potentially toxic dose in patients less than 6 years: greater than 0.5 mg/kg
Indication: Sedative/Muscle Relaxant
Age: greater than 12 years
Dose: Oral – 0.12-0.8 mg/kg/day
Frequency: divided every 6-8 hours
Note: by mouth (oral); Potentially toxic dose in patients less than 6 years: greater than 0.5 mg/kg

Renal Dose

Clinical InformationAdministration Information
Age: Adult
Condition: Renal impairment
Dose: Oral – Data not available
Note: No dose adjustment recommended unless administered for prolonged period; decrease dose in prolonged periods
Condition: Renal impairment
Dose: Rectal gel – Not studied
Note: Use caution
Administration
  • Take on empty stomach
  • Take 1 hour before or 2 hours after meals
Side Effect

Drug Interaction

Drug NameRisk Factors
Amprenavir, Ritonavir
May significantly enhance CNS depressant effect
Anesthetics, Narcotic analgesics, Antidepressants (Fluoxetine, Sertraline, Paroxetine, Citalopram, Escitalopram, Venlafaxine, Duloxetine), Antipsychotics (Haloperidol, Risperidone, Quetiapine, Olanzapine, Clozapine, Aripiprazole), Anxiolytics, Antiepileptics, Antihistamines (Diphenhydramine, Loratadine, Levocetirizine, Cetirizine, Fexofenadine, Hydroxyzine, Bilastin), Antihypertensive (Captopril, Enalapril, Lisinopril, Ramipril, Benazepril, Fosinopril, Quinapril, Perindopril, Losartan, Valsartan, Candesartan, Irbesartan, Telmisartan, Olmesartan, Propranolol, Metoprolol, Atenolol, Carvedilol, Bisoprolol, Nadolol, Amlodipine, Diltiazem, Verapamil, Nifedipine, Nicardipine, Hydrochlorothiazide, Chlorthalidone, Indapamide, Furosemide, Bumetanide, Torsemide, Spironolactone, Amiloride, Triamterene, Prazosin, Doxazosin, Terazosin, Clonidine, Methyldopa, Hydralazine, Minoxidil), Muscle Relaxants (Baclofen, Cyclobenzaprine, Tizanidine, Dantrolene) (e.g. tizanidine, baclofen), Nabilone
May enhance CNS depressant effect

Disease Interaction

Disease NameRisk Factors
Myasthenia Gravis
Can worsen muscle weakness
CNS Depression
Can increase sedation

Pregnancy

Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage
Store in a cool (below 25˚C temperature) and dry place protected from light.

Data Sources

Clinical & regulatory information on this page is compiled from the following government sources:

DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.