Medicine Overview
Adult Dose
| Clinical Information | Administration Information |
|---|---|
|
Indication: Benign gastric and duodenal ulceration Age: Adult Condition: Initial |
Dose: Oral – 300 mg daily at bedtime or 150 mg twice daily Frequency: once daily or twice daily Duration: 4-8 weeks Note: 300 mg twice daily for 4 weeks may be used in duodenal ulcer to improved healing. Maximum: 300 mg twice daily. Hepatic impairment: Dosage adjustment not necessary |
|
Indication: Benign gastric and duodenal ulceration Age: Adult Condition: Maintenance |
Dose: Oral – 150 mg Frequency: once daily at bedtime Note: Hepatic impairment: Dosage adjustment not necessary |
Child Dose
| Clinical Information | Administration Information |
|---|---|
|
Indication: Benign gastric and duodenal ulceration Age: 1 month to 16 years |
Dose: Oral – 4-8 mg/kg Frequency: daily in 2 divided doses Duration: 4-8 weeks Note: Maximum: 300 mg/day |
|
Indication: Benign gastric and duodenal ulceration Age: 1 month to 16 years Condition: Maintenance |
Dose: Oral – 2-4 mg/kg Frequency: once daily Note: Maximum: 150 mg/day |
Renal Dose
| Clinical Information | Administration Information |
|---|---|
|
Condition: Creatinine Clearance less than 50 |
Dose: Oral – 150 mg Frequency: daily at bedtime Note: adjust dose cautiously if necessary |
|
Condition: Renal Impairment |
Dose: Parenteral – 25 mg Note: Individual doses may be reduced |
Administration
- Can be taken with or without food
- For injection: Must be administered by healthcare professional
Side Effect
- Headache (3%)
- Abdominal pain
- Agitation
- Alopecia
- Confusion
- Constipation
- Diarrhea
- Dizziness
- Hypersensitivity reaction
- Nausea
- Vomiting
- Anemia
- Necrotizing enterocolitis in fetus or newborn
- Pancreatitis (rare)
- Thrombocytopenia (rare)
- Pancytopenia (rare)
- Agranulocytosis (rare)
- Acquired immune hemolytic anemia (rare)
- Arthralgia (rare)
- Anaphylaxis
- hypersensitivity reactions
Drug Interaction
Drug Interaction
| Drug Name | Risk Factors |
|---|---|
|
Propantheline bromide
|
Delayed absorption and increased peak serum concentration
|
|
Coumarin Anticoagulants (Warfarin, Heparin, Dabigatran, Rivaroxaban, Apixaban, Edoxaban), Theophylline, Diazepam, Propranolol
|
Minimally inhibits hepatic metabolism
|
Disease Interaction
Disease Interaction
| Disease Name | Risk Factors |
|---|---|
|
Porphyria
|
Can trigger acute attacks
|
Pregnancy
Pregnancy
Lactation
Special Use
Precaution
Overdose
Pharmacology
Storage
Store in a cool and dry place. protect from light.
Data Sources
Clinical & regulatory information on this page is compiled from the following government sources:
DISCLAIMER: This drug information content is provided for informational purposes only and is not intended to be a substitute for professional medical advice, diagnosis, or treatment. Patients should always consult their physician with any questions regarding a medical condition and to obtain medical advice and treatment.